Structure-based design, synthesis and in vitro characterization of potent 17β-hydroxysteroid dehydrogenase type 1 inhibitors based on 2-substitutions of estrone and d-homo-estrone.
Autor(en):
Möller, G. ; Deluca, D. ; Gege, C. ; Rosinus, A. ; Kowalik, D. ; Peters, O. ; Droescher, P. ; Elger, W. ; Adamski, J. ; Hillisch, A.